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Agonism
Opioid
mu-activity
delta activity
kappa activity
Common Name
Strong
Morphine
mu agonism
mu agonism
mu agonism
Duramorph
Heroin
mu agonism
mu agonism
mu agonism
Smack, H, Harry
Methadone
mu agonism
at high doses
at high doses
Dolophine
Hydromorphone
mu agonism
at high doses
at high doses
Dilaudid
Meperidine
mu agonism
at high doses
at high doses
Demerol
Fentanyl
mu agonism
at high doses
at high doses
Sublimaze
Alfentanil
mu agonism
at high doses
at high doses
Alfenta
Sufentanil
mu agonism
at high doses
at high doses
Sufenta
Moderate to Weak
Oxycodone
mu agonism
at high doses
at high doses
OxyContin
Hydrocodone
mu agonism
at high doses
at high doses
Vicodin
Codeine
mu agonism
at high doses
at high doses
Tylenol #3
Propoxyphene
mu agonism
at high doses
at high doses
Darvocet
Dextromethorphan
mu agonism
at high doses
at high doses
Robitussin DM
Diphenoxylate
mu agonism
at high doses
at high doses
Lomotil
Difenoxin
mu agonism
at high doses
at high doses
Motofen
Loperamide
mu agonism
at high doses
at high doses
Imodium AD
Mixed agonist/antagonist
Nalbuphine
mu agonism
no activity
mu agonism
Nubain
Pentazocine
partial agonist
no activity
mu agonism
Talwin
Butorphanol
partial agonist
no activity
mu agonism
Stadol
Buprenorphine
partial agonist
no activity
antagonist
Buprenex
Antagonists
Naloxone
antagonist
antagonist
antagonist
Narcan
Naltrexone
antagonist
antagonist
antagonist
Revia

Related terms: partial opioid agonist, opioid antagonist

 

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